Highly diastereoselective asymmetric Mannich reactions of 1,3-dicarbonyls with acyl imines.

نویسندگان

  • Amal Ting
  • Sha Lou
  • Scott E Schaus
چکیده

[reaction: see text] The cinchona alkaloids catalyze direct asymmetric Mannich reactions of cyclic 1,3-dicarbonyl compounds with acyl imines to afford alpha-quaternary carbon-bearing reaction products in yields of up to 98%, a diastereomeric excess of 90% or greater, and enantioselectivities up to 99% ee. A model is proposed that accounts for both the observed diastereoselectivities and the enantioselectivities for the reactions.

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Highly enantio- and diastereoselective Mannich reactions of glycine Schiff bases with in situ generated N-Boc-imines catalyzed by a cinchona alkaloid thiourea.

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عنوان ژورنال:
  • Organic letters

دوره 8 10  شماره 

صفحات  -

تاریخ انتشار 2006